SCHEMBL9038552

SCHEMBL9038552

CCn1c(=O)[nH]c2nccc(NC(C)C)c2c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 7/20 0.45
ADORA2A P29274 5/20 0.45
PDE4A P27815 4/20 0.45
PDE4C Q08493 4/20 0.45
PDE4D Q08499 4/20 0.45
CYP1A2 P05177 2/20 0.40
ADORA3 P0DMS8 5/20 0.40
ADORA2B P29275 5/20 0.40
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCND2 P30279 1/20 0.37
CCND3 P30281 1/20 0.37
HSD17B13 Q7Z5P4 1/20 0.36
PDE7A Q13946 3/20 0.36
PDE7B Q9NP56 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
UTS2R Q9UKP6 1/20 0.34
PARG Q86W56 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040427 0.82 ADORA2A (0.41) ADORA2AADORA3ADORA2BADORA1
SCHEMBL9038556 0.81 PDE4B (0.44) PDE4BADORA2APDE4APDE4CPDE4D
SCHEMBL9038149 0.78 ADORA2A (0.49) PDE4BADORA2APDE4APDE4CPDE4D
SCHEMBL9037741 0.77 ADORA2B (0.40) PDE4BADORA2APDE4APDE4CPDE4D
SCHEMBL9038040 0.75 PDE4B (0.43) PDE4BADORA2APDE4APDE4CPDE4D
SCHEMBL9039306 0.73 PDE4B (0.43) PDE4BADORA2APDE4APDE4CPDE4D
SCHEMBL9039080 0.72 ADORA2A (0.46) ADORA2AADORA3ADORA2BMEN1KMT2A
SCHEMBL9037748 0.72 AURKA (0.39) UTS2R
SCHEMBL9037826 0.69 KMT2A (0.50) ADORA3MEN1KMT2A
SCHEMBL1713392 0.69 FEN1 (0.60) PDE4BADORA2APDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696590-A1 Pyrido[2,3-d]pyrimidine derivatives, their preparation and their use as anti-asthma agents NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-02-14 EP disclosed