SCHEMBL9040443

SCHEMBL9040443

O=C1c2cnccc2CNc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.53
MAOB P27338 2/20 0.53
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
JAK2 O60674 1/20 0.42
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CCNT1 O60563 1/20 0.37
CCNT2 O60583 1/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37
CDK9 P50750 1/20 0.37
CCNA1 P78396 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11474110 0.83 CA12 (0.59) MAOAMAOBCA12CA9JAK2
SCHEMBL30704654 0.80 CA12 (0.46) MAOAMAOBCA12CA9JAK2
SCHEMBL4053483 0.76 CES1 (0.61) MAOAMAOBALDH1A1CYP11B1CYP11B2
SCHEMBL17108096 0.76 JAK2 (0.54) MAOAMAOBCA12CA9JAK2
SCHEMBL148437 0.73 CA12 (0.55) MAOAMAOBCA12CA9JAK2
SCHEMBL18533306 0.73 S100A4 (0.46) MAOAMAOBCA12CA9JAK2
SCHEMBL3066734 0.73 MAOA (0.87) MAOAMAOBGAANPSR1HSD17B10
Hydrochloric Acid SCHEMBL7086048 0.72 CA12 (0.53) MAOAMAOBCA12CA9JAK2
SCHEMBL9201794 0.71 MAOA (0.48) MAOAMAOBCA12CA9JAK2
SCHEMBL11660603 0.71 MAOB (0.55) MAOAMAOBGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0347831-B1 Pyridine derivatives and intermediates thereof KYOWA HAKKO KOGYO KK (JP) 1996-12-11 EP disclosed
US-4971964-A INHIBITORS OF THROMBOXANE SYNTHASE, CARDIOVASCULAR DISORDERS, ANTIINFLAMMATORU AGENTS, CANCER KYOWA HAKKO KOGYO CO., LTD. (JP) 1990-11-20 US disclosed
EP-0347831-A2 Pyridine derivatives and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1989-12-27 EP disclosed