SCHEMBL904310

SCHEMBL904310

COc1ccc2c(c1)CC(c1ccccc1)c1c-2[nH]c2ccc(OC)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA4 P22748 2/20 0.53
CA6 P23280 2/20 0.53
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 2/20 0.47
MAPT P10636 2/20 0.47
KMT2A Q03164 2/20 0.47
HSD17B10 Q99714 2/20 0.47
HPGD P15428 2/20 0.47
MAPKAPK2 P49137 3/20 0.45
ABCG2 Q9UNQ0 1/20 0.43
TSHR P16473 1/20 0.42
GFER P55789 1/20 0.42
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
GSK3B P49841 1/20 0.42
CDK5 Q00535 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10111840 0.84 HTR2C (0.40) CA1CA2CA4CA6HTR6
SCHEMBL904324 0.80 CA1 (0.50) CA1CA2CA4CA6ALDH1A1
SCHEMBL904332 0.74 SLC6A2 (0.46) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL9146594 0.73 CYP19A1 (0.63) CA1CA2ALDH1A1ABCG2TSHR
SCHEMBL5612189 0.70 MAPKAPK2 (0.43) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL5708478 0.70 CA1 (0.69) CA1CA2CA4CA6MAPKAPK2
SCHEMBL7132711 0.70 MAPK10 (0.64) CA1CA2CA4CA6ALDH1A1
SCHEMBL5708473 0.69 CA1 (0.55) CA1CA2CA4CA6ALDH1A1
SCHEMBL8946305 0.69 CA1 (0.73) CA1CA2CA4CA6ALDH1A1
SCHEMBL12301264 0.69 CA1 (0.78) CA1CA2CA4CA6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041227-A1 TETRACYCLIC HETEROCYCLE COMPOUNDS FOR TREATING HEPATITIS C VIRAL INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed