SCHEMBL904332

SCHEMBL904332

COc1ccc2c(c1)CC(c1ccccc1)c1c-2n(C)c2ccc(OC)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
SLC6A3 Q01959 2/20 0.46
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
HPGD P15428 2/20 0.45
MAPT P10636 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
MEN1 O00255 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45
NTRK1 P04629 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP19A1 P11511 3/20 0.40
DRD2 P14416 2/20 0.39
DRD1 P21728 1/20 0.39
DRD5 P21918 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904323 0.85 DRD2 (0.39) DRD2DRD1DRD5DRD3
SCHEMBL904313 0.81 DRD1 (0.39) ALDH1A1KDM4EHPGDSMN1; SMN2DRD1
SCHEMBL904319 0.81 NR1H2 (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1KDM4E
SCHEMBL904310 0.74 CA1 (0.53) SLC6A2SLC6A4SLC6A3ALDH1A1KDM4E
SCHEMBL9146594 0.72 CYP19A1 (0.63) SLC6A2SLC6A4SLC6A3ALDH1A1CYP19A1
SCHEMBL17697978 0.69 DRD2 (0.56) ALDH1A1KDM4EHPGDMAPTL3MBTL1
SCHEMBL1990706 0.69 DRD1 (0.55) ALDH1A1KDM4EHPGDMAPTL3MBTL1
SCHEMBL12601843 0.68 KDM4E (0.47) ALDH1A1KDM4EHPGDMAPTL3MBTL1
SCHEMBL1987539 0.67 DRD2 (0.53) ALDH1A1KDM4EHPGDMAPTL3MBTL1
SCHEMBL1986645 0.67 KDM4E (0.49) ALDH1A1KDM4EHPGDMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012041227-A1 TETRACYCLIC HETEROCYCLE COMPOUNDS FOR TREATING HEPATITIS C VIRAL INFECTION MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed