SCHEMBL9043333

SCHEMBL9043333

C[C@@](N)(C(=O)O)c1ccc(OCCOc2ccc3ccccc3c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.54
PPARG P37231 3/20 0.54
PPARD Q03181 3/20 0.54
KDM4E B2RXH2 4/20 0.53
ALDH1A1 P00352 1/20 0.53
MAPK1 P28482 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
PTPN7 P35236 1/20 0.51
CPT2 P23786 1/20 0.51
CPT1A P50416 1/20 0.51
CPT1B Q92523 1/20 0.51
HDAC1 Q13547 1/20 0.46
NPC1 O15118 2/20 0.46
MAPT P10636 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PKM P14618 1/20 0.45
AGXT P21549 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL514964 0.82 CYP1A2 (0.51) PPARAPTPN7MAPTPKM
SCHEMBL4755686 0.82 CYP1A2 (0.51) PPARAPTPN7MAPTPKM
SCHEMBL5970098 0.82 CYP1A2 (0.51) PPARAPTPN7MAPTPKM
SCHEMBL9042927 0.82 KDM4E (0.53) PPARAPPARGPPARDKDM4EALDH1A1
SCHEMBL28137765 0.77 PPARA (0.79) PPARAPPARGKDM4EALDH1A1MAPK1
SCHEMBL9335358 0.77 GPBAR1 (0.60)
SCHEMBL9232872 0.77 PKM (0.59) PPARGKDM4ENPC1MAPTRAB9A
SCHEMBL9232775 0.77 PKM (0.59) PPARGKDM4ENPC1MAPTRAB9A
SCHEMBL9232869 0.77 PKM (0.59) PPARGKDM4ENPC1MAPTRAB9A
SCHEMBL2177291 0.77 KDM4E (0.77) PPARAPPARGPPARDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512352-B1 Substituted carboxylic acid derivatives HOFFMANN LA ROCHE (CH) 1996-03-27 EP claimed
EP-0512352-B1 Substituted carboxylic acid derivatives HOFFMANN LA ROCHE (CH) 1996-03-27 EP disclosed
US-5344843-A Carnitine acryltransferase enzyme inhibitors as antiischemic agents and for cardiovascular disorders HOFFMAN-LA ROCHE INC. (US) 1994-09-06 US disclosed
EP-0512352-A2 Substituted carboxylic acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-11-11 EP disclosed