SCHEMBL9044262

SCHEMBL9044262

CC(N)C(=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
TSHR P16473 3/20 0.63
CES2 O00748 1/20 0.62
CES1 P23141 1/20 0.62
SLC6A2 P23975 1/20 0.60
CHRNB4 P30926 1/20 0.60
CHRNA3 P32297 1/20 0.60
SLC6A3 Q01959 1/20 0.60
TP53 P04637 1/20 0.60
KMO O15229 1/20 0.57
PRSS1 P07477 1/20 0.55
PRSS2 P07478 1/20 0.55
PRSS3 P35030 1/20 0.55
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
MAPT P10636 3/20 0.51
HTT P42858 1/20 0.51
RAB9A P51151 1/20 0.51
POLB P06746 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3844160 0.87 ALDH1A1 (0.67) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL29408207 0.87 ALDH1A1 (0.67) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL2599194 0.85 ALDH1A1 (0.65) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL2599404 0.85 ALDH1A1 (0.65) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL11064019 0.84 TSHR (0.64) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL9423190 0.84 ALDH1A1 (0.63) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL3801805 0.84 ALDH1A1 (0.63) ALDH1A1TSHRCES2CES1SLC6A2
Isobutane SCHEMBL6119723 0.82 TSHR (0.87) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL27914715 0.81 CES2 (0.68) ALDH1A1TSHRCES2CES1SLC6A2
SCHEMBL6400030 0.81 TP53 (0.61) ALDH1A1TSHRCES2CES1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0471358-B1 Fluoroethylcamptothecin derivatives KYORIN SEIYAKU KK (JP) 1996-05-08 EP disclosed
EP-0325247-B1 CAMPTOTHECIN DERIVATIVES AND PROCESS FOR PREPARING SAME KABUSHIKI KAISHA YAKULT HONSHA (JP) 1993-05-19 EP disclosed
EP-0471358-A1 Fluoroethylcamptothecin derivatives KYORIN PHARMACEUTICAL CO., LTD. (JP) 1992-02-19 EP disclosed
US-5061800-A ANTITUMOR AGENTS KABUSHIKI KAISHA YAKULT HONSHA (JP) 1991-10-29 US disclosed
EP-0325247-A1 Camptothecin derivatives and process for preparing same KABUSHIKI KAISHA YAKULT HONSHA (JP) 1989-07-26 EP disclosed