SCHEMBL9044285

SCHEMBL9044285

COC(=O)c1ccc(C#Cn2cnc3nc(NC(=O)C(C)(C)C)cc-3c2O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 3/20 0.38
ADORA1 P30542 1/20 0.36
PTPN11 Q06124 1/20 0.35
MAPT P10636 3/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9045602 0.90 ADORA1 (0.36) NPC1RAB9ASMN1; SMN2KDM4EADORA1
SCHEMBL9045445 0.89 ADORA1 (0.38) KDM4EADORA1CYP1A2CYP2C9CYP2C19
SCHEMBL9046427 0.88 ADORA1 (0.38) NPC1RAB9AADORA1MAPTCYP1A2
SCHEMBL9046822 0.88 ADORA1 (0.38) ADORA1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL9046114 0.88 ADORA1 (0.46) NPC1RAB9ASMN1; SMN2ADORA1CYP1A2
SCHEMBL9471023 0.83 KMT2A (0.43) RAB9ASMN1; SMN2KDM4EPTPN11MAPT
SCHEMBL9044777 0.82 ADORA1 (0.38) ADORA1ABL1
SCHEMBL9047678 0.81 MAPK14 (0.34) RAB9AKDM4EADORA1ALDH1A1HPGD
SCHEMBL9049865 0.80 CA2 (0.37) KDM4EHPGDCA12CA1CA2
SCHEMBL9044312 0.79 ADORA1 (0.39) NPC1RAB9AADORA1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed