SCHEMBL9045602

SCHEMBL9045602

COc1ccc(C#Cn2cnc3nc(NC(=O)C(C)(C)C)cc-3c2O)cc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ADORA3 P0DMS8 10/20 0.36
NPC1 O15118 2/20 0.35
TP53 P04637 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
ALDH1A1 P00352 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
HSP90AA1 P07900 1/20 0.35
ADORA2B P29275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044285 0.90 NPC1 (0.38) ADORA1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL9045445 0.89 ADORA1 (0.38) ADORA1LMNAADORA3TP53KDM4E
SCHEMBL9046822 0.88 ADORA1 (0.38) ADORA1LMNAADORA3
SCHEMBL9046427 0.88 ADORA1 (0.38) ADORA1LMNAADORA3NPC1RAB9A
SCHEMBL9046114 0.88 ADORA1 (0.46) ADORA1LMNANPC1TP53RAB9A
SCHEMBL9044777 0.82 ADORA1 (0.38) ADORA1
SCHEMBL9047678 0.80 MAPK14 (0.34) ADORA1L3MBTL1RAB9AALDH1A1KDM4E
SCHEMBL9044312 0.79 ADORA1 (0.39) ADORA1NPC1RAB9A
SCHEMBL9471269 0.79 APP (0.39) LMNANPC1TP53RAB9ASMN1; SMN2
SCHEMBL9049865 0.78 CA2 (0.37) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0432677-B1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives UNIV PRINCETON (US) 1996-03-06 EP disclosed
US-5344932-A N-(pyrrolo(2,3-d)pyrimidin-3-ylacyl)-glutamic acid derivatives TRUSTEES OF PRINCETON UNIVERSITY (US) 1994-09-06 US disclosed
US-5248775-A Pyrrolo(2,3-d)pyrimidines THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1993-09-28 US disclosed
EP-0432677-A1 N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-06-19 EP disclosed