SCHEMBL9045289

SCHEMBL9045289

Nc1nccnc1C(=O)N1CCCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
DPP4 P27487 1/20 0.48
PIM1 P11309 2/20 0.47
PIM3 Q86V86 2/20 0.47
PIM2 Q9P1W9 2/20 0.47
KDM4E B2RXH2 1/20 0.46
HPGD P15428 6/20 0.45
ALDH1A1 P00352 5/20 0.43
GAA P10253 1/20 0.41
HSD11B1 P28845 1/20 0.41
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PRKCI P41743 2/20 0.40
ATR Q13535 2/20 0.40
PRKDC P78527 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22840303 0.82 APOBEC3A (0.55) DPP4HPGDALDH1A1SMN1; SMN2
SCHEMBL7455826 0.77 PIM1 (0.52) KMT2APIM1PIM3KDM4EHPGD
SCHEMBL9044008 0.77 DPP4 (0.48) DPP4PIM1PIM3PIM2HPGD
SCHEMBL7522157 0.76 PIM1 (0.54) KMT2APIM1PIM3KDM4EHPGD
SCHEMBL11786826 0.75 KMT2A (0.47) KMT2APIM1PIM3PIM2KDM4E
SCHEMBL28382554 0.74 NAPRT (0.56) KMT2AKDM4EHPGDALDH1A1GAA
SCHEMBL7452732 0.74 PIM1 (0.49) KMT2APIM1PIM3PIM2KDM4E
SCHEMBL28326660 0.73 NAPRT (0.54) KMT2AKDM4EHPGDALDH1A1GAA
SCHEMBL9053116 0.71 HPGD (0.40) KMT2AHPGDALDH1A1MEN1
SCHEMBL9193063 0.71 SPR (0.67) KMT2APIM1KDM4EHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743944-A1 AZACYCLIC DERIVATIVES SmithKline Beecham Farmaceutici S.p.A. (IT) 1996-11-27 EP disclosed
WO-1995021843-A1 AZACYCLIC DERIVATIVES SMITHKLINE BEECHAM FARMACEUTICI S.P.A. (IT) 1995-08-17 WO disclosed
US-3954753-A SEDATIVES, MUSCLE RELAXANTS, ANTICONVULSANTS HOFFMANN-LA ROCHE INC. (US) 1976-05-04 US disclosed