SCHEMBL9047784

SCHEMBL9047784

CCOC(=O)c1ccc(-c2ccc3cc4c(cc3c2)C(C)(C)CCC4(C)C)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.67
RARA P10276 10/20 0.67
RARG P13631 7/20 0.67
PDK2 Q15119 1/20 0.49
RXRA P19793 2/20 0.46
KCNH2 Q12809 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
PDGFRB P09619 1/20 0.46
PDGFRA P16234 1/20 0.46
CYP3A4 P08684 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ESR1 P03372 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
ESR2 Q92731 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CYP26A1 O43174 1/20 0.44
CYP26B1 Q9NR63 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10959462 0.89 RARA (0.68) RARBRARARARGRXRACYP26A1
SCHEMBL9117300 0.85 RARB (0.54) RARBRARARARGPDK2RXRA
SCHEMBL9051570 0.85 RARB (0.56) RARBRARARARGPDK2RXRA
SCHEMBL8659260 0.85 RARA (0.54) RARBRARARARGPDGFRBPDGFRA
SCHEMBL9119758 0.84 RARB (0.53) RARBRARARARGPDK2RXRA
SCHEMBL9051778 0.84 RARB (0.53) RARBRARARARGPDK2RXRA
SCHEMBL8657242 0.83 RARA (0.50) RARBRARARARGPDK2RXRA
SCHEMBL9051144 0.83 RARB (0.53) RARBRARARARGPDK2RXRA
SCHEMBL9050623 0.83 RARB (0.52) RARBRARARARGRXRA
SCHEMBL9120469 0.83 RARB (0.52) RARBRARARARGPDK2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995033745-A9 NOVEL COMPOUNDS USEFUL IN MODULATING GENE EXPRESSION OF RETINOID RESPONSIVE GENES AND/OR HAVING ANTI-AP-1 ACTIVITY 1996-01-18 WO disclosed
WO-1995033745-A2 NOVEL COMPOUNDS USEFUL IN MODULATING GENE EXPRESSION OF RETINOID RESPONSIVE GENES AND/OR HAVING ANTI-AP-1 ACTIVITY SRI INTERNATIONAL (US) 1995-12-14 WO disclosed