SCHEMBL9048124

SCHEMBL9048124

CS(=O)(=O)c1ccc(-n2ccc(-c3ccc(F)cc3)n2)cc1

nearest known ligand 0.65

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.65
PTGS1 P23219 3/20 0.65
FAAH O00519 1/20 0.52
KCNH2 Q12809 1/20 0.52
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
AOC3 Q16853 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9048815 0.87 PTGS2 (0.64) PTGS2PTGS1CA1CA2
SCHEMBL9047084 0.86 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL9047072 0.86 PTGS2 (0.65) PTGS2PTGS1FAAHKCNH2
SCHEMBL9040666 0.86 PTGS2 (0.57) PTGS2PTGS1CA1CA2
SCHEMBL8423922 0.86 MELK (0.59) PTGS2PTGS1
SCHEMBL9046017 0.83 PTGS2 (0.51) PTGS2PTGS1FAAHKCNH2
SCHEMBL9038989 0.83 PTGS2 (0.67) PTGS2PTGS1CA1CA2
SCHEMBL9047083 0.82 PTGS2 (0.57) PTGS2PTGS1KCNH2CA1CA2
SCHEMBL9038455 0.82 PTGS2 (0.50) PTGS2PTGS1CA1CA2
SCHEMBL8421061 0.78 PTGS2 (0.88) PTGS2PTGS1AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731796-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP disclosed
WO-1995015318-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed