SCHEMBL9048815

SCHEMBL9048815

Cc1ccc(-c2ccn(-c3ccc(S(C)(=O)=O)cc3)n2)cc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.64
PTGS1 P23219 8/20 0.64
CYP2C9 P11712 1/20 0.52
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA5A P35218 1/20 0.49
CA9 Q16790 1/20 0.49
CA5B Q9Y2D0 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9040666 0.87 PTGS2 (0.57) PTGS2PTGS1CA1CA2
SCHEMBL8423922 0.87 MELK (0.59) PTGS2PTGS1CA12CA9
SCHEMBL9047084 0.87 PTGS2 (0.55) PTGS2PTGS1CA12CA9
SCHEMBL9048124 0.87 PTGS2 (0.65) PTGS2PTGS1CA1CA2
SCHEMBL9047072 0.87 PTGS2 (0.65) PTGS2PTGS1
SCHEMBL9046017 0.85 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL9038989 0.85 PTGS2 (0.67) PTGS2PTGS1CA1CA2CA5A
SCHEMBL9038455 0.83 PTGS2 (0.50) PTGS2PTGS1CA12CA1CA2
SCHEMBL9047083 0.83 PTGS2 (0.57) PTGS2PTGS1CA12CA1CA2
SCHEMBL13801011 0.78 HTT (0.50) PTGS2PTGS1CYP2C9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731796-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP disclosed
WO-1995015318-A1 1,3,5-TRISUBSTITUTED PYRAZOLE COMPOUNDS FOR TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed