SCHEMBL9045019

SCHEMBL9045019

NC1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)cn3CCF)C1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 7/20 0.71
ALDH1A1 P00352 6/20 0.70
DRD3 P35462 1/20 0.58
KDM4E B2RXH2 4/20 0.55
HPGD P15428 4/20 0.55
HSD17B10 Q99714 4/20 0.55
LMNA P02545 3/20 0.55
BRD4 O60885 1/20 0.55
TSHR P16473 1/20 0.55
HTT P42858 1/20 0.55
CYP2J2 P51589 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
KMT2A Q03164 2/20 0.54
MEN1 O00255 1/20 0.54
NPC1 O15118 1/20 0.54
PRKD3 O94806 1/20 0.53
PIM1 P11309 1/20 0.53
GSK3A P49840 1/20 0.53
GSK3B P49841 1/20 0.53
IRAK1 P51617 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9048236 0.90 TOP1 (0.71) TOP1ALDH1A1DRD3KDM4EHPGD
Hydrochloric Acid SCHEMBL8571733 0.89 TOP1 (0.70) TOP1ALDH1A1DRD3KDM4EHPGD
SCHEMBL30626291 0.89 ALDH1A1 (0.71) TOP1ALDH1A1DRD3KDM4EHPGD
SCHEMBL9750142 0.85 ALDH1A1 (0.69) TOP1ALDH1A1DRD3KDM4EHPGD
SCHEMBL9045127 0.84 TOP1 (0.61) TOP1ALDH1A1DRD3KDM4EHPGD
SCHEMBL5571927 0.84 ALDH1A1 (0.71) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL5571931 0.84 ALDH1A1 (0.71) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL5571992 0.84 ALDH1A1 (0.71) TOP1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2854967 0.83 ALDH1A1 (0.72) TOP1ALDH1A1DRD3KDM4EHPGD
SCHEMBL2856476 0.83 ALDH1A1 (0.82) ALDH1A1DRD3KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360258-B1 Amino acid quinoline and naphthyridine derivatives ABBOTT LAB (US) 1996-08-14 EP disclosed
US-5057523-A Water soluble bactericide ABBOTT LABORATORIES (US) 1991-10-15 US disclosed
EP-0360258-A2 Amino acid quinoline and naphthyridine derivatives ABBOTT LABORATORIES (US) 1990-03-28 EP disclosed