SCHEMBL9048398

SCHEMBL9048398

O=C(O)Cn1c(=S)c2cc(Cl)ccc2n(Cc2ccc(Br)cc2F)c1=O

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 8/20 0.69
AKR1A1 P14550 3/20 0.69
AKR1B10 O60218 4/20 0.52
PTGDR2 Q9Y5Y4 2/20 0.41
OPRM1 P35372 1/20 0.40
TRAP1 Q12931 2/20 0.40
TBXA2R P21731 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90B1 P14625 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056716 0.90 AKR1B1 (0.78) AKR1B1AKR1A1AKR1B10PTGDR2MEN1
SCHEMBL10488007 0.88 AKR1B1 (0.85) AKR1B1AKR1A1AKR1B10PTGDR2OPRM1
SCHEMBL9046869 0.87 AKR1B1 (0.53) AKR1B1AKR1A1AKR1B10OPRM1TRAP1
SCHEMBL9049383 0.87 AKR1B1 (0.60) AKR1B1AKR1A1AKR1B10PTGDR2TBXA2R
Zenarestat SCHEMBL30583313 0.82 AKR1B1 (1.00) AKR1B1AKR1A1AKR1B10OPRM1TRAP1
Zenarestat SCHEMBL29688249 0.82 AKR1B1 (1.00) AKR1B1AKR1A1AKR1B10OPRM1TRAP1
Zenarestat SCHEMBL48959 0.82 AKR1B1 (1.00) AKR1B1AKR1A1AKR1B10OPRM1TRAP1
SCHEMBL9046879 0.81 AKR1B1 (0.55) AKR1B1AKR1A1AKR1B10TRAP1TBXA2R
SCHEMBL9048160 0.77 AKR1B1 (0.52) AKR1B1AKR1A1AKR1B10TBXA2RMEN1
SCHEMBL9046143 0.77 AKR1A1 (0.59) AKR1B1AKR1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456835-B1 QUINAZOLINE-3-ALKANOIC ACID DERIVATIVE, SALT THEREOF, AND PRODUCTION THEREOF KYORIN SEIYAKU KK (JP) 1996-05-15 EP disclosed
US-5234928-A Inhibit platelet aggregation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1993-08-10 US disclosed
EP-0456835-A1 QUINAZOLINE-3-ALKANOIC ACID DERIVATIVE, SALT THEREOF, AND PRODUCTION THEREOF KYORIN PHARMACEUTICAL CO., LTD. (JP) 1991-11-21 EP disclosed