SCHEMBL9048770

SCHEMBL9048770

C/C=C/C(C1=C(O)CC(c2ccccc2)(c2ccccc2)OC1=O)c1cccc(C)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LDHA P00338 6/20 0.37
LDHB P07195 6/20 0.37
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OPRK1 P41145 2/20 0.35
OPRL1 P41146 2/20 0.35
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ACP3 P15309 1/20 0.34
HSD11B1 P28845 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
CYP3A4 P08684 2/20 0.31
CYP2C19 P33261 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP2C9 P11712 1/20 0.31
HSD17B2 P37059 1/20 0.31
SLC6A9 P48067 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6604874 0.76 LDHA (0.42) LDHALDHBOPRM1OPRL1CYP3A4
SCHEMBL6605852 0.68 LDHA (0.41) LDHALDHBLMNANPSR1HSD11B1
SCHEMBL9026061 0.68 LDHA (0.43) LDHALDHBOPRM1OPRD1OPRK1
SCHEMBL6172935 0.66 KDM4E (0.30)
SCHEMBL6175498 0.65 LDHA (0.34) LDHAOPRD1ALDH1A1
SCHEMBL6603297 0.62 LDHA (0.58) LDHALDHB
SCHEMBL6604700 0.62 LDHA (0.58) LDHALDHB
SCHEMBL7441906 0.62 LDHA (0.38) LDHALDHB
SCHEMBL6604488 0.62 LDHA (0.52) LDHALDHBOPRM1OPRD1ALDH1A1
SCHEMBL6174563 0.62 LDHA (0.35) LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729464-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP claimed
EP-0729464-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed