SCHEMBL9049337

SCHEMBL9049337

Cc1[nH]c2ccccc2c1C(=O)[C@H]1CCc2[nH]cnc2C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.48
ADRA2A P08913 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
SLC6A4 P31645 1/20 0.48
OPRK1 P41145 1/20 0.48
HTR2B P41595 1/20 0.48
KCNH2 Q12809 1/20 0.48
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
RAB9A P51151 4/20 0.44
NPC1 O15118 2/20 0.44
NR4A2 P43354 1/20 0.41
ALDH1A1 P00352 5/20 0.41
KMT2A Q03164 5/20 0.41
LMNA P02545 3/20 0.41
MITF O75030 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271791 1.00 HTR3A (0.48) HTR3AADRA2AADRA2BADRA2CSLC6A4
Fumaric Acid SCHEMBL9050456 0.94 HTR3A (0.43) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL16585577 0.91 HTR3A (0.58) HTR3AADRA2AADRA2BADRA2CSLC6A4
Fumaric Acid SCHEMBL9050462 0.86 HTR3A (0.52) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL9048273 0.83 HTR3A (0.43) HTR3AADRA2AADRA2BADRA2CSLC6A4
Fumaric Acid SCHEMBL9050460 0.81 SIRT1 (0.40) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL3175918 0.80 CYP2C19 (0.56) HTR3AADRA2AADRA2BADRA2CSLC6A4
Fumaric Acid SCHEMBL9050432 0.80 HTR3A (0.40) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL3180338 0.79 HTR3A (0.55) HTR3AADRA2AADRA2BADRA2CSLC6A4
SCHEMBL3180342 0.79 HTR3A (0.55) HTR3AADRA2AADRA2BADRA2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP claimed