SCHEMBL9049869

SCHEMBL9049869

O=C(O)Cn1c(=O)[nH]c2ccc(Cl)cc2c1=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.60
CA9 Q16790 1/20 0.60
ALDH1A1 P00352 3/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
POLB P06746 1/20 0.56
PKM P14618 1/20 0.56
KDM4E B2RXH2 1/20 0.48
HPGD P15428 1/20 0.48
CHEK1 O14757 1/20 0.47
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
JAK2 O60674 1/20 0.47
MAP4K4 O95819 1/20 0.47
ABL1 P00519 1/20 0.47
NTRK1 P04629 1/20 0.47
LCK P06239 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
MET P08581 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31161048 0.84 CA9 (0.55) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL10084481 0.83 KDM4E (0.50) ALDH1A1MEN1KMT2APOLBKDM4E
SCHEMBL640508 0.82 CBX7 (0.58) CA12CA9
SCHEMBL9045056 0.82 ALDH1A1 (0.57) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL11009308 0.81 CA12 (0.61) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL31160880 0.80 KDM4E (0.45) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL11008112 0.79 CA12 (0.59) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL3311524 0.79 ALDH1A1 (0.73) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL8987779 0.78 CA12 (0.57) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL7655193 0.76 CA12 (0.58) CA12CA9ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4688756-A1 QUINAZOLINE DIONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2026-02-11 EP disclosed
WO-2024206345-A1 QUINAZOLINE DIONE COMPOUNDS AND USES THEREOF EDGEWISE THERAPEUTICS, INC. (US) 2024-10-03 WO disclosed
EP-0456835-B1 QUINAZOLINE-3-ALKANOIC ACID DERIVATIVE, SALT THEREOF, AND PRODUCTION THEREOF KYORIN SEIYAKU KK (JP) 1996-05-15 EP disclosed
US-5234928-A Inhibit platelet aggregation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1993-08-10 US disclosed
EP-0456835-A1 QUINAZOLINE-3-ALKANOIC ACID DERIVATIVE, SALT THEREOF, AND PRODUCTION THEREOF KYORIN PHARMACEUTICAL CO., LTD. (JP) 1991-11-21 EP disclosed