SCHEMBL9050464

SCHEMBL9050464

CCOC(=O)c1ccc(-c2cc(CN3CCCC3)c3cc4c(cc3c2)C(C)(C)CCC4(C)C)cc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
RARA P10276 5/20 0.47
RARB P10826 5/20 0.47
RARG P13631 2/20 0.47
ALDH1A1 P00352 5/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
HPGD P15428 2/20 0.39
PDK2 Q15119 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
PTGER4 P35408 1/20 0.38
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9050569 0.86 RARB (0.56) RARARARBRARG
SCHEMBL9049309 0.86 RARB (0.52) RARARARBRARGALDH1A1MAPT
SCHEMBL9051247 0.85 RARA (0.53) RARARARBRARGPDK2
SCHEMBL9050339 0.83 RARB (0.49) KCNH2HRH3RARARARBRARG
SCHEMBL9117300 0.82 RARB (0.54) RARARARBRARGESR1ESR2
SCHEMBL9051118 0.82 RARA (0.51) RARARARBRARGMAPTPDK2
SCHEMBL9119758 0.81 RARB (0.53) KCNH2HRH3RARARARBRARG
SCHEMBL9051778 0.81 RARB (0.53) RARARARBRARGESR1ESR2
SCHEMBL9051144 0.81 RARB (0.53) RARARARBRARGPDK2MAPK1
SCHEMBL9050623 0.80 RARB (0.52) RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995033745-A9 NOVEL COMPOUNDS USEFUL IN MODULATING GENE EXPRESSION OF RETINOID RESPONSIVE GENES AND/OR HAVING ANTI-AP-1 ACTIVITY 1996-01-18 WO disclosed
WO-1995033745-A2 NOVEL COMPOUNDS USEFUL IN MODULATING GENE EXPRESSION OF RETINOID RESPONSIVE GENES AND/OR HAVING ANTI-AP-1 ACTIVITY SRI INTERNATIONAL (US) 1995-12-14 WO disclosed