SCHEMBL9050600

SCHEMBL9050600

O=C(C1CCc2[nH]cnc2C1)N1CCc2ccccc2C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.55
ALDH1A1 P00352 5/20 0.52
TSHR P16473 2/20 0.52
MAPK1 P28482 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPT P10636 2/20 0.48
HTT P42858 2/20 0.48
POLB P06746 1/20 0.48
KDM4E B2RXH2 3/20 0.47
HPGD P15428 3/20 0.47
LMNA P02545 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
GAA P10253 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
RIPK1 Q13546 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9050604 0.91 KEAP1 (0.55) KEAP1ALDH1A1TSHRMAPK1KMT2A
SCHEMBL1023584 0.82 TSHR (0.59) ALDH1A1TSHRMAPK1KMT2AMAPT
SCHEMBL1023583 0.82 TSHR (0.59) ALDH1A1TSHRMAPK1KMT2AMAPT
Hydrochloric Acid SCHEMBL1023299 0.81 TSHR (0.57) ALDH1A1TSHRMAPK1KMT2AMAPT
Hydrochloric Acid SCHEMBL9050997 0.81 TSHR (0.57) ALDH1A1TSHRMAPK1KMT2AMAPT
SCHEMBL3182983 0.80 HPGD (0.41) ALDH1A1TSHRKMT2AHTTHPGD
Hydrochloric Acid SCHEMBL9051125 0.79 HPGD (0.40) ALDH1A1TSHRKMT2AHTTHPGD
SCHEMBL6418657 0.78 KDM4E (0.51) KEAP1ALDH1A1TSHRKMT2AMAPT
Fumaric Acid SCHEMBL9051209 0.77 TSHR (0.52) ALDH1A1TSHRMAPK1KMT2AMAPT
SCHEMBL9052644 0.76 ALOX15 (0.49) ALDH1A1TSHRKMT2AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381422-B1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMA CO LTD (JP) 1996-10-23 EP disclosed
US-5496942-A 5-HT3-RECEPTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-03-05 US disclosed
US-5344927-A 5-HT3 antagonist YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0381422-A1 Tetrahydrobenzimidazole derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1990-08-08 EP disclosed