SCHEMBL9050810

SCHEMBL9050810

CCCCCc1c(C(N)=O)cc(N)c(N)c1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.42
BRD4 O60885 2/20 0.42
IKBKB O14920 2/20 0.41
DHFR P00374 1/20 0.40
DPP4 P27487 1/20 0.40
MEN1 O00255 1/20 0.40
NR1I2 O75469 1/20 0.40
LMNA P02545 1/20 0.40
CHRM2 P08172 1/20 0.40
CYP3A4 P08684 1/20 0.40
ADRA2A P08913 1/20 0.40
MAPT P10636 1/20 0.40
OPRK1 P41145 1/20 0.40
HTR2B P41595 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KMT2A Q03164 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CNR2 P34972 1/20 0.39
ALOX15 P16050 4/20 0.39
GRK6 P43250 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27318113 0.82 BRD4 (0.42) GCGRBRD4IKBKBDPP4MEN1
SCHEMBL9051709 0.79 GCGR (0.44) GCGRBRD4DHFRDPP4MEN1
SCHEMBL8027233 0.76 IKBKB (0.43) BRD4IKBKBMEN1NR1I2LMNA
SCHEMBL28621722 0.73 DHFR (0.49) GCGRDHFR
SCHEMBL4301700 0.73 GCGR (0.43) GCGRBRD4DPP4MEN1NR1I2
SCHEMBL10903924 0.72 CYP3A4 (0.48) GCGRMEN1NR1I2LMNACHRM2
SCHEMBL5370893 0.71 CYP3A4 (0.53) MEN1NR1I2LMNACHRM2CYP3A4
SCHEMBL11323683 0.70 RARB (0.49) GCGRRARB
SCHEMBL2882017 0.70 DHFR (0.52) GCGRDHFRCNR2
SCHEMBL7060341 0.70 DHFR (0.52) GCGRDHFRCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722439-A1 HIV PROTEASE INHIBITORS AGOURON PHARMACEUTICALS, INC. (US) 1996-07-24 EP disclosed