SCHEMBL9051708

SCHEMBL9051708

COc1cc(OC)nc(OC(C(=O)O)C(O)(c2ccccc2)C(F)(F)F)n1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 20/20 0.75
EDNRA P25101 20/20 0.75
NR1I2 O75469 1/20 0.51
KCNE1 P15382 1/20 0.51
KCNQ1 P51787 1/20 0.51
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9051649 0.87 EDNRB (0.61) EDNRBEDNRA
SCHEMBL9369015 0.83 EDNRB (0.76) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL6776490 0.83 EDNRB (0.76) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL6776058 0.82 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1
Darusentan SCHEMBL1068546 0.82 EDNRB (1.00) EDNRBEDNRANR1I2KCNE1KCNQ1
Darusentan SCHEMBL795084 0.82 EDNRB (1.00) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL1067551 0.81 EDNRB (0.73) EDNRBEDNRANR1I2KCNE1KCNQ1
SCHEMBL7071036 0.81 EDNRB (1.00) EDNRBEDNRA
SCHEMBL9052058 0.80 EDNRB (0.53) EDNRBEDNRA
SCHEMBL12228356 0.80 EDNRB (0.71) EDNRBEDNRANR1I2KCNE1KCNQ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996000219-A1 PYRIMIDINYL- AND TRIAZINYL-OXY AND THIO-3-HALOALKYL-PROPIONIC ACID DERIVATIVES AS HERBICIDES CIBA-GEIGY AG (CH) 1996-01-04 WO disclosed