SCHEMBL9052228

SCHEMBL9052228

O=C(O)Nc1ccc(N2CCN(CCC3CCc4ccccc43)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.47
DRD3 P35462 4/20 0.47
HTR1A P08908 3/20 0.47
LMNA P02545 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
DRD4 P21917 3/20 0.45
DRD1 P21728 2/20 0.45
POLB P06746 1/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
ADRA1D P25100 1/20 0.45
HTR2A P28223 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
HTR2B P41595 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402811 0.84 DRD2 (0.46) DRD2DRD3HTR1ADRD4DRD1
SCHEMBL7405539 0.83 ALDH1A1 (0.53) DRD2DRD3HTR1ALMNADRD4
SCHEMBL7403486 0.83 DRD2 (0.50) DRD2DRD3HTR1ADRD4DRD1
SCHEMBL7404378 0.82 MAPT (0.52) DRD2HTR1ADRD4POLBHTR2A
Hydrochloric Acid SCHEMBL8185523 0.82 ALDH1A1 (0.52) DRD2DRD3HTR1ALMNADRD4
Hydrochloric Acid SCHEMBL7401818 0.81 MAPT (0.51) DRD2HTR1ADRD4POLBHTR2A
SCHEMBL27524409 0.78 DRD2 (0.69) DRD2DRD3HTR1ADRD4DRD1
SCHEMBL7401374 0.78 DRD2 (0.48) DRD2DRD3HTR1ADRD4DRD1
SCHEMBL7397854 0.78 DRD4 (0.68) DRD2HTR1ADRD4HTR2AADRA1A
Hydrochloric Acid SCHEMBL8185604 0.77 DRD4 (0.67) DRD2HTR1ADRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737189-A1 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF CNS AND CARDIOVASCULAR DISORDERS PHARMACIA & UPJOHN COMPANY (US) 1996-10-16 EP disclosed