SCHEMBL9052397

SCHEMBL9052397

[CH2]Cc1ccnc(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.38
PTGS2 P35354 3/20 0.38
HTR2B P41595 1/20 0.37
HTR5A P47898 1/20 0.37
TDO2 P48775 1/20 0.37
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
AURKA O14965 1/20 0.35
HSP90AA1 P07900 1/20 0.35
PRKACA P17612 1/20 0.35
ADORA2A P29274 1/20 0.35
KDM4E B2RXH2 3/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
ALOX15 P16050 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
MAPT P10636 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2494339 0.81 KDM4E (0.40) PTGS2HTR2BHTR5ATDO2PDE3B
SCHEMBL5309860 0.81 HTR2B (0.37) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL29986186 0.81 PTGS1 (0.46) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL27650879 0.81 PTGS1 (0.35) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL10584953 0.75 PTGS1 (0.41) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL2491635 0.73 ADORA2A (0.50) ADORA2AKDM4EL3MBTL1NPC1RAB9A
SCHEMBL996432 0.72 CCNA2 (0.45) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL10381277 0.72 HTR2B (0.41) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL321472 0.71 CCNA2 (0.44) PTGS1PTGS2HTR2BHTR5ATDO2
SCHEMBL10205841 0.71 PTGS1 (0.46) PTGS1PTGS2HTR2BHTR5ATDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004297-A9 SYNTHESIS AND USE OF AMINO ACID FLUORIDES AS PEPTIDE COUPLING REAGENTS 1996-05-02 WO disclosed