SCHEMBL9052939

SCHEMBL9052939

Nc1nccc(CC2CNCCO2)n1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.39
SLC6A4 P31645 4/20 0.39
SLC6A2 P23975 2/20 0.39
HTR2B P41595 2/20 0.39
SLC6A3 Q01959 2/20 0.39
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA2C P18825 1/20 0.39
HRH3 Q9Y5N1 3/20 0.38
HRH1 P35367 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR3A P46098 1/20 0.38
IRAK4 Q9NWZ3 6/20 0.37
KDR P35968 2/20 0.35
SYK P43405 2/20 0.35
NLRP3 Q96P20 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5624032 0.82 HTR2A (0.41) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL28029187 0.76 HTR2A (0.40) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL5338566 0.75 SLC6A2 (0.48) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL30637279 0.75 HTR2A (0.42) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL6616733 0.75 ADRB2 (0.39) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL27948442 0.74 PLAU (0.39) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL5346300 0.73 SLC6A2 (0.41) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL15416051 0.73 SLC6A2 (0.37) HTR2ASLC6A4SLC6A2HTR2BSLC6A3
SCHEMBL28798379 0.72 DRD2 (0.42)
SCHEMBL27854563 0.72 SLC6A2 (0.42) HTR2ASLC6A4SLC6A2HTR2BSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP claimed