SCHEMBL9052989

SCHEMBL9052989

CCc1cccc(C2(O)CCN(CCCC(=O)c3ccc(F)cc3)CC2)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.74
CYP3A4 P08684 3/20 0.72
CYP2D6 P10635 3/20 0.72
ABCB11 O95342 2/20 0.72
TSHR P16473 2/20 0.72
THPO P40225 2/20 0.72
MTOR P42345 2/20 0.72
EBP Q15125 2/20 0.72
SIGMAR1 Q99720 2/20 0.72
TP53 P04637 1/20 0.72
PKM P14618 1/20 0.72
MAPK1 P28482 1/20 0.72
PMP22 Q01453 2/20 0.71
KDM4E B2RXH2 1/20 0.71
SMN1; SMN2 Q16637 1/20 0.71
CYP1A2 P05177 2/20 0.64
HTR1A P08908 2/20 0.64
ADRA2A P08913 2/20 0.64
CHRM1 P11229 2/20 0.64
ADRA2B P18089 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9053428 0.91 DRD2 (0.74) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9053658 0.88 DRD2 (0.82) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9050989 0.88 DRD2 (0.77) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9053091 0.87 DRD2 (0.84) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9051330 0.85 DRD2 (0.77) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9053114 0.85 DRD2 (0.73) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL8986042 0.85 DRD2 (1.00) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9053173 0.84 DRD2 (0.82) DRD2CYP3A4CYP2D6ABCB11TSHR
Trifluperidol SCHEMBL120862 0.84 CYP3A4 (1.00) DRD2CYP3A4CYP2D6ABCB11TSHR
Trifluperidol SCHEMBL29710906 0.84 CYP3A4 (1.00) DRD2CYP3A4CYP2D6ABCB11TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002250-A1 HALOPERIDOL ANALOGS AND THE USE THEREOF ACEA PHARMACEUTICALS INC. (US) 1996-02-01 WO disclosed