SCHEMBL9053972

SCHEMBL9053972

COc1ccc(S(=O)(=O)N2CCOc3ccccc32)cc1-c1ccc[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.59
POLB P06746 1/20 0.54
KMT2A Q03164 5/20 0.49
MEN1 O00255 3/20 0.49
MAPT P10636 2/20 0.49
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
USP2 O75604 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP2C9 P11712 1/20 0.41
HTR6 P50406 1/20 0.40
LMNA P02545 1/20 0.40
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9058745 0.83 PDE4A (0.69) KMT2AMEN1MAPTPDE4APDE4B
SCHEMBL9054130 0.81 KMT2A (0.63) NPC1KMT2AMEN1MAPTPDE4A
SCHEMBL8541489 0.78 KDM4E (0.60) NPC1POLBUSP2GAAALDH1A1
SCHEMBL9053909 0.78 NPC1 (0.64) NPC1POLBKMT2AMEN1MAPT
SCHEMBL8540258 0.77 GPBAR1 (0.60) KMT2AMEN1USP2ALDH1A1LMNA
SCHEMBL8588242 0.77 GPBAR1 (0.56) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL8543576 0.76 MCOLN3 (0.58) GAAPKMALDH1A1LMNA
SCHEMBL14758405 0.75 NPC1 (1.00) NPC1POLBKMT2AMEN1MAPT
SCHEMBL8539014 0.74 L3MBTL1 (0.51) POLBUSP2ALDH1A1LMNA
SCHEMBL8544818 0.72 AKR1C3 (0.44) POLBMAPTCYP3A4USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0734378-A1 AMINOSULPHONYL-PHENYL-1H-PYRROLE DERIVATIVES, METHOD OF THEIR PREPARATION AND THEIR USE SMITHKLINE BEECHAM PLC (GB) 1996-10-02 EP disclosed
WO-1995016674-A1 AMINOSULPHONYL-PHENYL-1H-PYRROLE DERIVATIVES, METHOD OF THEIR PREPARATION AND THEIR USE SMITHKLINE BEECHAM PLC (GB) 1995-06-22 WO disclosed