SCHEMBL9054202

SCHEMBL9054202

CNC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@]2(O)C(C)(C)[C@]12O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.55
ADORA3 P0DMS8 5/20 0.52
PI4KA P42356 2/20 0.48
PI4K2B Q8TCG2 2/20 0.48
PI4K2A Q9BTU6 2/20 0.48
PI4KB Q9UBF8 2/20 0.48
ADORA2B P29275 4/20 0.45
TSHR P16473 4/20 0.44
KMT2A Q03164 3/20 0.44
ADORA1 P30542 3/20 0.44
HSP90AA1 P07900 2/20 0.44
HSP90B1 P14625 2/20 0.44
AHCY P23526 2/20 0.44
LMNA P02545 1/20 0.44
THRB P10828 1/20 0.44
BLM P54132 1/20 0.44
MAPK1 P28482 3/20 0.43
MEN1 O00255 2/20 0.43
DPP4 P27487 1/20 0.43
SLC28A1 O00337 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28156591 0.88 ADORA2A (0.64) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL19692161 0.88 ADORA2A (0.58) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL1078828 0.88 ADORA2A (0.64) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL11040343 0.88 ADORA2A (0.58) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL8943715 0.87 ADORA2A (0.57) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL5554234 0.86 ADORA2A (0.56) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL8943533 0.82 ADORA2A (0.53) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL8943541 0.82 ADORA2A (0.55) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL8943868 0.82 ADORA2A (0.53) ADORA2AADORA3PI4KAPI4K2BPI4K2A
SCHEMBL25408738 0.82 ADORA2A (0.52) ADORA2AADORA3PI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472181-B1 5-Amine substituted adenosine analogs as immunosuppressants MERRELL PHARMA INC (US) 1996-10-02 EP disclosed
EP-0358536-B1 Novel S-adenosyl methionine decarboxylase inhibitors MERRELL PHARMA INC (US) 1996-05-08 EP disclosed
US-5416076-A S-adenosyl methionine decarboxylase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1995-05-16 US disclosed
US-5308837-A 5'-amine substituted adenosine analogs as immunosuppressants MERRELL DOW PHARMACEUTICALS INC. (US) 1994-05-03 US disclosed
EP-0472181-A2 5-Amine substituted adenosine analogs as immunosuppressants MERRELL PHARMACEUTICALS INC. (US) 1992-02-26 EP disclosed
EP-0358536-A2 Novel S-adenosyl methionine decarboxylase inhibitors MERRELL PHARMACEUTICALS INC. (US) 1990-03-14 EP disclosed
EP-0351475-A1 S-Adenosylmethionine decarboxylase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1990-01-24 EP disclosed