SCHEMBL9054913

SCHEMBL9054913

CCOC(=O)O[C@@H]1CCCCN1C(=O)[C@H](CCCNc1ncc[nH]1)NS(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
ITGB3 P05106 2/20 0.40
ITGAV P06756 2/20 0.40
ITGA2B P08514 2/20 0.40
GAA P10253 2/20 0.39
ATM Q13315 1/20 0.39
HTR7 P34969 3/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
F2 P00734 3/20 0.37
ALOX15 P16050 2/20 0.37
MAPK1 P28482 1/20 0.37
TSHR P16473 2/20 0.37
POLB P06746 2/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 1/20 0.37
LMNA P02545 1/20 0.36
HTR6 P50406 2/20 0.36
PKLR P30613 1/20 0.36
CCR10 P46092 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9055193 0.94 ITGB3 (0.39) ALDH1A1ITGB3ITGAVITGA2BF2
SCHEMBL9056467 0.91 ITGB3 (0.43) ALDH1A1ITGB3ITGAVITGA2BGAA
SCHEMBL9055882 0.91 ITGB3 (0.38) ALDH1A1ITGB3ITGAVITGA2BF2
SCHEMBL9056658 0.91 ITGB3 (0.40) ITGB3ITGAVITGA2BF2CCR10
SCHEMBL9055118 0.89 ITGB3 (0.42) ITGB3ITGAVITGA2BF2CCR10
SCHEMBL9055094 0.88 ITGB3 (0.40) ITGB3ITGAVITGA2BF2CCR10
SCHEMBL9058970 0.86 F2 (0.54) F2
SCHEMBL9055638 0.86 ITGB3 (0.41) ITGB3ITGAVITGA2BF2CCR10
SCHEMBL9062251 0.86 F2 (0.48) ITGB3ITGAVITGA2BF2
SCHEMBL9056463 0.85 F2 (0.44) ITGB3ITGAVITGA2BGAAHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002517-A1 SUBSTITUTED ARYLSULFONAMIDES, THEIR PREPARATION AND USE AS THROMBIN-INHIBITING MEDICAMENTS DR. KARL THOMAE GMBH (DE) 1996-02-01 WO disclosed