SCHEMBL9056467

SCHEMBL9056467

O=C(O)O[C@@H]1CCCCN1C(=O)[C@H](CCCNc1ncc[nH]1)NS(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.43
ITGAV P06756 5/20 0.43
ITGA2B P08514 5/20 0.43
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTR7 P34969 1/20 0.40
TSHR P16473 2/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
F2 P00734 5/20 0.38
ALDH1A1 P00352 3/20 0.38
POLB P06746 1/20 0.38
RECQL P46063 1/20 0.38
LMNA P02545 1/20 0.37
MCOLN3 Q8TDD5 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9055638 0.92 ITGB3 (0.41) ITGB3ITGAVITGA2BF2
SCHEMBL9054913 0.91 ALDH1A1 (0.43) ITGB3ITGAVITGA2BMAPTGAA
SCHEMBL9056463 0.89 F2 (0.44) ITGB3ITGAVITGA2BMAPTGAA
SCHEMBL9055686 0.89 ITGB3 (0.43) ITGB3ITGAVITGA2BF2
SCHEMBL9055294 0.88 ITGB3 (0.46) ITGB3ITGAVITGA2BF2
SCHEMBL9058855 0.87 ITGB3 (0.43) ITGB3ITGAVITGA2BF2
SCHEMBL9060440 0.85 F2 (0.49) ITGB3ITGAVITGA2BF2
SCHEMBL9058775 0.85 F2 (0.56) ITGB3ITGAVITGA2BF2
SCHEMBL9055193 0.85 ITGB3 (0.39) ITGB3ITGAVITGA2BF2ALDH1A1
SCHEMBL9057064 0.84 F2 (0.51) ITGB3ITGAVITGA2BMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002517-A1 SUBSTITUTED ARYLSULFONAMIDES, THEIR PREPARATION AND USE AS THROMBIN-INHIBITING MEDICAMENTS DR. KARL THOMAE GMBH (DE) 1996-02-01 WO disclosed