SCHEMBL9056045

SCHEMBL9056045

CC(=O)OC1CC(=O)c2c(n(Cc3ccccc3)c3ccccc23)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
ABCB1 P08183 1/20 0.43
P2RX4 Q99571 1/20 0.43
CHRM2 P08172 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
CHRM1 P11229 1/20 0.42
DRD1 P21728 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA1A P35348 1/20 0.42
OPRM1 P35372 1/20 0.42
DRD3 P35462 1/20 0.42
SLC6A3 Q01959 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27470535 0.89 HDAC6 (0.44) HDAC1HDAC6HTR3EHTR3BHTR3A
SCHEMBL9056969 0.82 CA1 (0.48) HDAC1HDAC6HTR3EHTR3BHTR3A
SCHEMBL9055755 0.80 CHRM2 (0.50) HDAC1HDAC6CHRM2HTR1AADRA2A
SCHEMBL27470534 0.78 HDAC6 (0.46) HDAC1HDAC6HTR3EHTR3BHTR3A
SCHEMBL8387262 0.78 HDAC1 (0.47) HDAC1HDAC6P2RX4CHRM2HTR1A
SCHEMBL27470537 0.77 P2RX4 (0.50) HDAC1HDAC6P2RX4CHRM2HTR1A
SCHEMBL9056678 0.77 HDAC1 (0.49) HDAC1HDAC6HTR3EHTR3BHTR3A
SCHEMBL27489205 0.72 CA1 (0.46) HDAC1HDAC6HTR3EHTR3BHTR3A
SCHEMBL9057318 0.71 HDAC6 (0.48) HDAC1HDAC6CHRM2HTR1AADRA2A
SCHEMBL30480036 0.71 HDAC1 (0.70) HDAC1HDAC6P2RX4CHRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1166169-A Heterocyclic compounds, useful as allosteric effectors at muscarinic receptors SANKYO CO (JP) 1997-11-26 CN disclosed
WO-1996003377-A1 HETEROCYCLIC COMPOUNDS, USEFUL AS ALLOSTERIC EFFECTORS AT MUSCARINIC RECEPTORS SANKYO COMPANY, LIMITED (JP) 1996-02-08 WO disclosed