SCHEMBL9056280

SCHEMBL9056280

COc1ccc(C=NNC(=O)OC(C)(C)C)c(OC(C)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.54
MAPT P10636 8/20 0.50
KMT2A Q03164 6/20 0.50
MEN1 O00255 5/20 0.50
ALDH1A1 P00352 4/20 0.49
LMNA P02545 2/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 2/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
POLB P06746 1/20 0.47
MIF P14174 1/20 0.47
PKM P14618 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
RECQL P46063 1/20 0.46
ALOX12 P18054 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18692791 0.90 KDM4E (0.62) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL18692790 0.90 KDM4E (0.62) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL9056279 0.89 KDM4E (0.52) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL915761 0.81 MAPT (0.53) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL2488962 0.76 MIF (0.74) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL2488965 0.76 MIF (0.74) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL1573371 0.74 KDM4E (0.67) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL1573369 0.74 KDM4E (0.67) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL9055047 0.74 ALDH1A1 (0.71) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL18704469 0.73 MAPT (0.67) KDM4EMAPTKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996012706-A1 NOVEL ACID PYRAZOLE AND PYRAZOLONE DERIVATIVES FOR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS ROUSSEL UCLAF (FR) 1996-05-02 WO disclosed