SCHEMBL9057654

SCHEMBL9057654

CC(=O)OCCCn1cc(C2=C(c3c[nH]c4ccccc34)C(=O)N(C)C2=O)c2ccccc21

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 1/20 0.72
CCNT1 O60563 2/20 0.61
CDK9 P50750 2/20 0.61
PRKACA P17612 10/20 0.59
PRKACG P22612 10/20 0.59
PRKACB P22694 10/20 0.59
CDK4 P11802 4/20 0.59
CCND1 P24385 4/20 0.59
CAMK2D Q13557 4/20 0.56
CCNB2 O95067 3/20 0.56
CDK1 P06493 3/20 0.56
CCNB1 P14635 3/20 0.56
CCNB3 Q8WWL7 3/20 0.56
SIRT2 Q8IXJ6 2/20 0.56
SIRT1 Q96EB6 2/20 0.56
PIM1 P11309 2/20 0.56
GSK3B P49841 2/20 0.56
CCNE2 O96020 2/20 0.56
CCNE1 P24864 2/20 0.56
CDK2 P24941 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9374625 0.88 RPS6KB1 (0.77) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL8317356 0.82 RPS6KB1 (0.50) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL7199461 0.82 PRKACA (0.81) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL28101193 0.80 RPS6KB1 (0.74) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL14041797 0.77 PRKD1 (0.67) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL7195523 0.77 CCNT1 (0.81) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL8162860 0.76 CCNT1 (0.53) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL3945882 0.75 SIRT2 (1.00) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL30958473 0.75 SIRT2 (1.00) RPS6KB1CCNT1CDK9PRKACAPRKACG
SCHEMBL9376063 0.74 PRKACA (0.68) RPS6KB1CCNT1CDK9PRKACAPRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018765-A1 INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO claimed
WO-1996004906-A1 COMPOUNDS FOR THE TREATMENT OF RESTENOSIS THE WELLCOME FOUNDATION LIMITED (GB) 1996-02-22 WO disclosed
WO-1993018765-A1 INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO disclosed