SCHEMBL9057736

SCHEMBL9057736

O=C(O)c1ccc(C=Cc2cccnc2OCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A1 P22736 1/20 0.50
NR4A2 P43354 1/20 0.50
NR4A3 Q92570 1/20 0.50
SRD5A2 P31213 2/20 0.47
PPIA P62937 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.45
PLA2G4B P0C869 1/20 0.45
GSK3B P49841 1/20 0.44
BACE1 P56817 1/20 0.44
MAOB P27338 2/20 0.44
PTGER1 P34995 1/20 0.43
PTGER4 P35408 1/20 0.43
PTGER3 P43115 1/20 0.43
PTGER2 P43116 1/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
PSMD14 O00487 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326381 0.88 HTT (0.49) PPIAGSK3BBACE1MAOBKMT2A
SCHEMBL8325277 0.88 HTT (0.49) PPIAGSK3BBACE1MAOBKMT2A
SCHEMBL8318304 0.85 NR4A1 (0.48) NR4A1NR4A2NR4A3SRD5A2PPIA
SCHEMBL8318302 0.85 NR4A1 (0.48) NR4A1NR4A2NR4A3SRD5A2PPIA
SCHEMBL7774919 0.82 PTGER1 (0.64) NR4A1NR4A2NR4A3SRD5A2PTGER1
SCHEMBL7767009 0.78 NR4A2 (0.81) NR4A1NR4A2NR4A3SRD5A2ABCG2
SCHEMBL8676414 0.76 KMT2A (0.48) PPIAPTGER1PTGER4PTGER3PTGER2
SCHEMBL4035249 0.75 CCNB2 (0.47) MAOBPTGER1PTGER4PTGER3PTGER2
SCHEMBL8676412 0.75 PTGER4 (0.47) PTGER1PTGER4PTGER3PTGER2KDM4E
SCHEMBL8322839 0.74 PTGER4 (0.57) NR4A1NR4A2NR4A3SRD5A2PPIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed