SCHEMBL9057753

SCHEMBL9057753

CC(=O)N1CCc2ccc(C)cc2CC1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.58
MCHR1 Q99705 3/20 0.49
PTAFR P25105 2/20 0.49
HRH3 Q9Y5N1 1/20 0.49
BAZ2B Q9UIF8 1/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
KCNA1 Q09470 2/20 0.45
KCNAB1 Q14722 2/20 0.45
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HDAC6 Q9UBN7 1/20 0.42
RORC P51449 1/20 0.42
AKR1C3 P42330 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7992940 0.90 NOTUM (0.65) NOTUMBAZ2BRAB9ANPC1ALDH1A1
SCHEMBL12287671 0.90 NOTUM (0.65) NOTUMHRH3BAZ2BRAB9ANPC1
SCHEMBL7275642 0.82 ESR2 (0.56) NOTUMPTAFRHRH3
SCHEMBL6952918 0.81 NOTUM (0.59) NOTUMMCHR1PTAFRHRH3BAZ2B
SCHEMBL2310027 0.81 NR1H2 (0.57) NOTUMMCHR1PTAFRHRH3BAZ2B
SCHEMBL29295623 0.81 NOTUM (0.53) NOTUMPTAFRHRH3BAZ2BRAB9A
SCHEMBL3440214 0.81 RAB9A (0.53) NOTUMMCHR1HRH3RAB9ANPC1
SCHEMBL11068898 0.81 NOTUM (0.59) NOTUMMCHR1PTAFRALDH1A1
SCHEMBL12013933 0.80 NOTUM (0.53) NOTUMMCHR1HRH3BAZ2BRAB9A
SCHEMBL3440261 0.79 ALDH1A1 (0.61) NOTUMMCHR1HRH3ALDH1A1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed
EP-0229510-B1 SULFINYL AND SULFONYL SUBSTITUTED-3-BENZAZEPINES SMITHKLINE BEECHAM CORPORATION (US) 1990-06-06 EP disclosed
US-4824839-A Sulfinyl and sulfonyl substituted 2,3,4,5 tetrahydro-1H-3-benzazepines and their use in treating gastrointestinal motility disorders SMITHKLINE BECKMAN CORPORATION (US) 1989-04-25 US disclosed
EP-0229510-A1 Sulfinyl and sulfonyl substituted-3-benzazepines SMITHKLINE BEECHAM CORPORATION (US) 1987-07-22 EP disclosed