SCHEMBL9057829

SCHEMBL9057829

CC(=O)N1CCN(CCN2C=Cc3cc(S(N)(=O)=O)sc3S2)CC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.37
LOX P28300 1/20 0.37
CA2 P00918 8/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.33
DRD3 P35462 1/20 0.33
THRB P10828 3/20 0.33
HRH3 Q9Y5N1 1/20 0.32
SIGMAR1 Q99720 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9115082 0.85 KDM1A (0.34) KDM1ALOXL3MBTL1ALDH1A1DRD3
SCHEMBL9058827 0.83 CA2 (0.47) CA2HRH3CA12CA1CA9
SCHEMBL8950325 0.78 CA2 (0.38) KDM1ALOXCA2L3MBTL1ALDH1A1
SCHEMBL9057323 0.72 CA2 (0.43) CA2CA12CA1CA9
SCHEMBL9058021 0.71 CA2 (0.34) CA2
SCHEMBL9058428 0.71 CA2 (0.34) CA2CA12CA1CA9
SCHEMBL9058203 0.70 CA2 (0.44) CA2
SCHEMBL9058842 0.69 CA2 (0.47) CA2
SCHEMBL9058179 0.65 CA2 (0.42) CA2HRH3CA12CA1CA9
SCHEMBL23823660 0.64 CYP1A2 (0.64) KDM1AL3MBTL1ALDH1A1DRD3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022099-A1 OPHTHALMIC COMPOSITIONS FOR TREATING GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-25 WO disclosed
WO-1995019981-A1 THIENOTHIAZINE SULFONAMIDE DERIVATIVES PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS CARBONIC ANHYDRASE INHIBITORS ALCON LABORATORIES, INC. (US) 1995-07-27 WO disclosed