SCHEMBL9058306

SCHEMBL9058306

COc1ccc(N2C=Cc3cc(S(N)(=O)=O)sc3S2)cc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA2 P00918 18/20 0.44
CA1 P00915 7/20 0.41
CA9 Q16790 4/20 0.41
CA12 O43570 3/20 0.41
CA4 P22748 2/20 0.34
CA5A P35218 2/20 0.34
CA5B Q9Y2D0 2/20 0.34
PTGS2 P35354 2/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9057297 0.78 MAPT (0.40) CA2CA1CA9CA12
SCHEMBL8950515 0.74 CA2 (0.46) CA2CA1CA9CA12CA4
SCHEMBL9058849 0.71 CA2 (0.39) CA2CA1CA9CA12CA4
SCHEMBL9057323 0.69 CA2 (0.43) CA2CA1CA9CA12CA4
SCHEMBL9058842 0.66 CA2 (0.47) CA2CA4
SCHEMBL9058428 0.66 CA2 (0.34) CA2CA1CA9CA12CA4
SCHEMBL9057333 0.65 CA2 (0.47) CA2CA1CA9CA12CA4
SCHEMBL9828441 0.63 CA2 (0.50) CA2CA1CA9CA12PTGS2
SCHEMBL2089350 0.62 CA2 (1.00) CA2
SCHEMBL2087596 0.62 CA2 (1.00) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996022099-A1 OPHTHALMIC COMPOSITIONS FOR TREATING GLAUCOMA ALCON LABORATORIES, INC. (US) 1996-07-25 WO disclosed
WO-1995019981-A1 THIENOTHIAZINE SULFONAMIDE DERIVATIVES PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS CARBONIC ANHYDRASE INHIBITORS ALCON LABORATORIES, INC. (US) 1995-07-27 WO disclosed