SCHEMBL9828441

SCHEMBL9828441

COc1ccc(Sc2sc(S(N)(=O)=O)cc2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA2 P00918 14/20 0.50
CA1 P00915 4/20 0.45
CA9 Q16790 4/20 0.45
CA12 O43570 3/20 0.45
DHFR P00374 1/20 0.42
PTGS2 P35354 2/20 0.41
PTGS1 P23219 1/20 0.41
STS P08842 1/20 0.39
PTGIR P43119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829393 0.82 CA2 (0.44) CA2CA1CA9CA12DHFR
SCHEMBL11125385 0.75 CA2 (0.45) CA2CA1CA9CA12
SCHEMBL9827840 0.74 CA2 (0.58) CA2CA1CA9CA12PTGS2
SCHEMBL958207 0.70 CA2 (0.46) CA2CA1CA9CA12
SCHEMBL9424674 0.69 CA2 (0.42) CA2
SCHEMBL9828861 0.67 FBP1 (0.45) CA2CA1CA9CA12DHFR
SCHEMBL2087596 0.67 CA2 (1.00) CA2
SCHEMBL2089350 0.67 CA2 (1.00) CA2
SCHEMBL5808577 0.66 GUSB (0.44) CA2CA1CA9CA12
SCHEMBL8105269 0.66 PTGS2 (0.48) CA2CA1CA9CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0295049-B1 THIOPHENE SULFONAMIDE ANTIGLAUCOMA AGENTS MERCK & CO. INC. (US) 1991-10-09 EP disclosed
US-4847289-A Thiophene sulfonamide antiglaucoma agents MERCK & CO., INC. (US) 1989-07-11 US disclosed
EP-0295049-A2 Thiophene sulfonamide antiglaucoma agents MERCK & CO. INC. (US) 1988-12-14 EP disclosed