SCHEMBL9059236

SCHEMBL9059236

Cc1cc(NNN)ccc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
IDO1 P14902 1/20 0.44
ALDH1A1 P00352 5/20 0.44
RAB9A P51151 8/20 0.42
NPC1 O15118 6/20 0.42
MAPT P10636 5/20 0.42
KMT2A Q03164 3/20 0.41
PKM P14618 1/20 0.41
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 2/20 0.40
POLB P06746 2/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
LMNA P02545 2/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL849744 0.83 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
Hydrochloric Acid SCHEMBL3464344 0.81 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL10981978 0.79 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL5840849 0.76 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
Hydrochloric Acid SCHEMBL28901909 0.74 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL19339699 0.74 CYP1A2 (0.49) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL879876 0.71 CYP3A4 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL8292659 0.71 RAB9A (0.53) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL12883522 0.71 CYP1A2 (0.46) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL6831800 0.71 ALDH1A1 (0.59) CYP1A2CYP3A4CYP2C9CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996019477-A1 TETRACYCLIC SPIRO COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-06-27 WO disclosed