SCHEMBL9059800

SCHEMBL9059800

CN(C)C(=O)C1CCN(C(N)=Nc2ccccc2-c2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 2/20 0.43
SIGMAR1 Q99720 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
PDK2 Q15119 2/20 0.39
NPSR1 Q6W5P4 1/20 0.37
CYP2D6 P10635 1/20 0.37
KDM4E B2RXH2 1/20 0.36
PRMT5 O14744 2/20 0.36
WDR77 Q9BQA1 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9059944 0.81 SIGMAR1 (0.48) SIGMAR1SMN1; SMN2NPSR1KDM4EALDH1A1
SCHEMBL9059900 0.80 SIGMAR1 (0.49) SIGMAR1SMN1; SMN2
SCHEMBL9059465 0.78 SIGMAR1 (0.45) SIGMAR1
SCHEMBL9060099 0.78 SIGMAR1 (0.47) SIGMAR1CYP2D6
SCHEMBL9059786 0.76 SIGMAR1 (0.46) SIGMAR1KDM4EKMT2A
SCHEMBL9061357 0.76 SIGMAR1 (0.60) SIGMAR1SMN1; SMN2NPSR1CYP2D6KDM4E
SCHEMBL9059245 0.75 SIGMAR1 (0.44) SIGMAR1SMN1; SMN2PDK2
SCHEMBL9059436 0.75 SIGMAR1 (0.44) SIGMAR1KMT2A
SCHEMBL9059367 0.73 SIGMAR1 (0.46) SIGMAR1ALDH1A1
SCHEMBL9311235 0.73 SIGMAR1 (0.46) SIGMAR1SMN1; SMN2KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996017612-A1 USE OF SUBSTITUTED PHENYLAMIDINE AND PHENYLGUANIDINE COMPOUNDS FOR THE TREATMENT OF CEREBRAL AND CARDIAC ISCHAEMIA, CONVULSION AND SICKLE CELL ANAEMIA KNOLL AKTIENGESELLSCHAFT (DE) 1996-06-13 WO disclosed
EP-0536151-B1 ORTHOSUBSTITUTED BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM BOOTS CO PLC (GB) 1994-09-14 EP disclosed
US-5302720-A Biphenyl-substituted guanidine derivatives useful as hypoglycaemic agents THE BOOTS COMPANY (GB) 1994-04-12 US disclosed