SCHEMBL9060269

SCHEMBL9060269

COc1ccc(C=Cc2ccc(OC(F)F)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 1/20 0.62
RELA Q04206 2/20 0.59
TRPA1 O75762 1/20 0.59
CYP1A2 P05177 3/20 0.57
CYP1A1 P04798 3/20 0.57
CYP1B1 Q16678 3/20 0.57
ESR1 P03372 2/20 0.57
PTGS2 P35354 2/20 0.57
TUBB4A P04350 2/20 0.57
TUBB P07437 2/20 0.57
TUBA3C P0DPH7 2/20 0.57
AHR P35869 2/20 0.57
TUBA1B P68363 2/20 0.57
TUBA4A P68366 2/20 0.57
TUBB4B P68371 2/20 0.57
TUBB3 Q13509 2/20 0.57
TUBB2A Q13885 2/20 0.57
TUBB8 Q3ZCM7 2/20 0.57
TUBA3E Q6PEY2 2/20 0.57
TUBA1A Q71U36 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2536970 0.87 CA1 (0.58) KDM4ECYP3A4LMNAALDH1A1NPC1
SCHEMBL9605427 0.84 CYP1A1 (0.69) CYP1A2CYP1A1CYP1B1ESR1PTGS2
SCHEMBL7793047 0.83 GRIN2D (0.53) NFE2L2CYP1A2PTGS2KDM4ECYP3A4
SCHEMBL7793053 0.83 GRIN2D (0.53) NFE2L2CYP1A2PTGS2KDM4ECYP3A4
SCHEMBL14950253 0.82 RELA (0.81) NFE2L2RELATRPA1CYP1A2CYP1A1
SCHEMBL4881152 0.82 RELA (0.81) NFE2L2RELATRPA1CYP1A2CYP1A1
SCHEMBL699457 0.82 RELA (0.81) NFE2L2RELATRPA1CYP1A2CYP1A1
SCHEMBL631998 0.82 RELA (0.81) NFE2L2RELATRPA1CYP1A2CYP1A1
SCHEMBL699458 0.82 RELA (0.81) NFE2L2RELATRPA1CYP1A2CYP1A1
SCHEMBL13790336 0.82 RELA (0.81) NFE2L2RELATRPA1CYP1A2CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5389292-A Liquid crystalline media having positive dielctric anisotropy, chemical, heat and radiation resistance, used as electro-optical displaying MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-14 US disclosed
CN-1023699-C Difluoromethyl compounds MERCK PATENT GMBH (DE) 1994-02-09 CN disclosed
EP-0381728-B1 DIFLUOROMETHYL COMPOUNDS MERCK PATENT GMBH (DE) 1993-12-08 EP disclosed
CN-1039797-A difluoromethyl compound MERCK PATENT GMBH (DE) 1990-02-21 CN disclosed