SCHEMBL9060469

SCHEMBL9060469

FC(F)(F)Oc1ccccc1CCOc1ncccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2J2 P51589 1/20 0.44
SLC6A3 Q01959 6/20 0.41
DRD2 P14416 5/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
SLC6A2 P23975 4/20 0.39
PHF8 Q9UPP1 1/20 0.39
SLC6A4 P31645 3/20 0.37
CYP2D6 P10635 2/20 0.37
KCNH2 Q12809 2/20 0.37
KCNN3 Q9UGI6 1/20 0.37
GRIN2B Q13224 3/20 0.36
GRIN1 Q05586 2/20 0.36
ABCB1 P08183 1/20 0.36
HTR1A P08908 1/20 0.36
HSD17B13 Q7Z5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9061838 0.84 EPHX2 (0.46) EPHX2CYP2C9CYP2J2SLC6A3DRD2
SCHEMBL2091568 0.78 SLC6A3 (0.49) EPHX2SLC6A3DRD2HDAC3HDAC1
SCHEMBL2091566 0.77 SLC6A3 (0.45) EPHX2SLC6A3DRD2HDAC3HDAC1
SCHEMBL5543073 0.76 FFAR4 (0.40) EPHX2SLC6A3DRD2HDAC3HDAC1
SCHEMBL6003155 0.74 SLC6A3 (0.43) EPHX2SLC6A3DRD2HDAC3HDAC1
SCHEMBL5164077 0.73 HDAC3 (0.64) EPHX2CYP2C9CYP2J2HDAC3HDAC1
SCHEMBL2097493 0.73 SLC6A3 (0.42) EPHX2SLC6A3DRD2HDAC3HDAC1
SCHEMBL2097495 0.73 SLC6A3 (0.42) EPHX2SLC6A3DRD2HDAC3HDAC1
SCHEMBL23881813 0.73 SLC6A3 (0.48) SLC6A3DRD2HDAC3HDAC1HDAC2
SCHEMBL2095128 0.73 SLC6A3 (0.47) SLC6A3DRD2HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5324449-A Substituted phenyl trifluoromethyl ethers MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-06-28 US disclosed
EP-0334911-B1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1993-02-10 EP disclosed
EP-0334911-A1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1989-10-04 EP disclosed