SCHEMBL9065338

SCHEMBL9065338

CCOCOc1cccc(Cl)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
DRD4 P21917 1/20 0.35
BTK Q06187 1/20 0.35
NCF1 P14598 1/20 0.35
CDK9 P50750 1/20 0.34
DYRK1A Q13627 1/20 0.34
DYRK2 Q92630 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
KCNH2 Q12809 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
GRM5 P41594 2/20 0.33
HTR7 P34969 1/20 0.33
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
KDM4E B2RXH2 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30271358 0.85 MAPK8 (0.49) MAPK8L3MBTL1DRD4BTKCDK9
SCHEMBL1671304 0.85 MAPK8 (0.49) MAPK8L3MBTL1DRD4BTKCDK9
SCHEMBL30436204 0.80 DRD4 (0.35) L3MBTL1DRD4CDK9DYRK1ADYRK2
SCHEMBL12483137 0.80 DRD4 (0.35) L3MBTL1DRD4CDK9DYRK1ADYRK2
SCHEMBL10910803 0.78 MCHR1 (0.42) MAPK8L3MBTL1DRD4CDK9DYRK1A
SCHEMBL10911295 0.76 MCHR1 (0.44) L3MBTL1CDK9DYRK1ADYRK2ALDH1A1
Ammonia Solution, Strong SCHEMBL2186005 0.76 MCHR1 (0.41) MAPK8L3MBTL1DRD4CDK9DYRK1A
SCHEMBL27852278 0.75 MCHR1 (0.45) CDK9DYRK1ADYRK2TSHRKCNH2
SCHEMBL7520131 0.74 MCHR1 (0.47) CDK9DYRK1ADYRK2TSHRKCNH2
SCHEMBL27852180 0.74 MCHR1 (0.47) CDK9DYRK1ADYRK2TSHRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486615-A Method of making asymmetric DE ring intermediates for the synthesis of camptothecin analogs NORTH CAROLINA STATE UNIVERSITY (US) 1996-01-23 US disclosed
US-5395939-A Method of making asymmetric de ring intermediates for the synthesis of camptothecin and camptothecin analogs NORTH CAROLINA STATE UNIVERSITY (US) 1995-03-07 US disclosed