SCHEMBL9065893

SCHEMBL9065893

Cc1c(NC(=O)c2[nH]nc(NC(=O)c3cc(N)nn3C)c2C)n[nH]c1C(=O)NCCC(=N)N

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRAS P01112 9/20 0.39
ESR1 P03372 9/20 0.39
ESR2 Q92731 9/20 0.39
TOP1 P11387 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HIF1A Q16665 1/20 0.39
BDKRB1 P46663 4/20 0.37
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038778 0.92 TOP1 (0.35) HRASESR1ESR2TOP1KDM4E
SCHEMBL9040554 0.85 HRAS (0.36) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL9038991 0.84 KDM4E (0.48) HRASESR1ESR2TOP1KDM4E
SCHEMBL9040894 0.83 HRAS (0.39) HRASESR1ESR2TOP1KDM4E
SCHEMBL9038376 0.82 HRAS (0.37) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL9037845 0.80 KDM4E (0.38) HRASESR1ESR2TOP1KDM4E
SCHEMBL8692462 0.79 HRAS (0.48) HRASESR1ESR2TOP1KDM4E
SCHEMBL9039671 0.79 BDKRB1 (0.38) HRASESR1ESR2TOP1KDM4E
SCHEMBL9037287 0.79 BDKRB1 (0.38) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL6613308 0.78 KDM4E (0.49) HRASESR1ESR2TOP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722446-A1 DISTAMYCIN A ANALOGUES AS ANTITUMOUR OR ANTIVIRAL AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 1996-07-24 EP disclosed
WO-1996005196-A1 DISTAMYCIN A ANALOGUES AS ANTITUMOUR OR ANTIVIRAL AGENTS PHARMACIA S.P.A. (IT) 1996-02-22 WO disclosed