SCHEMBL9068427

SCHEMBL9068427

C=CCc1c(C#N)cnc(N)c1C#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
CSNK1A1 P48729 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
HSD17B10 Q99714 4/20 0.35
ALOX15 P16050 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
IMPDH2 P12268 1/20 0.32
GAA P10253 2/20 0.31
HTT P42858 2/20 0.31
TSHR P16473 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28289900 0.78 USP7 (0.41) TP53CSNK1A1CLK4HSD17B10ALDH1A1
SCHEMBL8320187 0.75 MAPK1 (0.42) TP53CSNK1A1CLK4HSD17B10ALOX15
SCHEMBL9067611 0.74 TP53 (0.43) TP53CSNK1A1CLK4
SCHEMBL8321298 0.73 KDM4E (0.45) CSNK1A1CLK4HSD17B10ALDH1A1KDM4E
SCHEMBL10696235 0.72 TP53 (0.57) TP53CSNK1A1CLK4HSD17B10ALOX15
SCHEMBL11598649 0.72 TP53 (0.43) TP53CSNK1A1CLK4HSD17B10ALOX15
SCHEMBL8653737 0.71 KDM4E (0.37) HSD17B10ALOX15ALDH1A1KDM4EMAPT
SCHEMBL27883134 0.71 CSNK1A1 (0.47) TP53CSNK1A1CLK4KDM4EGAA
SCHEMBL11812461 0.70 MAPK1 (0.40) TP53HSD17B10ALOX15ALDH1A1KDM4E
SCHEMBL10690802 0.68 KDM4E (0.44) TP53CSNK1A1CLK4HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536724-A Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins SRI INTERNATIONAL (US) 1996-07-16 US disclosed