SCHEMBL10690802

SCHEMBL10690802

Cc1c(C#N)cnc(N)c1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.44
CSNK1A1 P48729 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
ABL1 P00519 1/20 0.40
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
HTT P42858 4/20 0.37
HSD17B10 Q99714 3/20 0.37
ADORA2A P29274 2/20 0.37
ADRA2A P08913 1/20 0.37
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
GRM6 O15303 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865549 0.87 ALDH1A1 (0.41) KDM4EALDH1A1CSNK1A1CLK4ABL1
SCHEMBL15894822 0.86 KDM4E (0.46) KDM4EALDH1A1ABL1NOS3NOS1
SCHEMBL3190550 0.83 CSNK1A1 (0.47) KDM4EALDH1A1CSNK1A1CLK4ABL1
SCHEMBL8650942 0.83 ALDH1A1 (0.38) KDM4EALDH1A1CSNK1A1CLK4ABL1
SCHEMBL2339904 0.82 CSNK1A1 (0.46) KDM4EALDH1A1CSNK1A1CLK4ABL1
SCHEMBL20489454 0.80 HTT (0.44) KDM4EALDH1A1CSNK1A1CLK4ABL1
SCHEMBL26194109 0.79 TSHR (0.37) KDM4EALDH1A1CSNK1A1CLK4HTT
SCHEMBL27883134 0.79 CSNK1A1 (0.47) KDM4ECSNK1A1CLK4ABL1HTT
SCHEMBL30937680 0.78 ALDH1A1 (0.43) KDM4EALDH1A1ABL1HTTHSD17B10
SCHEMBL8655458 0.78 ALDH1A1 (0.43) KDM4EALDH1A1ABL1NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4725687-A ANTITUMOR AGENTS; SIDE EFFECT REDUCTION; POTENCY SOUTHERN RESEARCH INSTITUTE (US) 1988-02-16 US disclosed