SCHEMBL9068436

SCHEMBL9068436

CCOC(=O)CC[C@H](NC(=O)c1ccc(C(C)c2cnc3nc(N)nc(N)c3c2C)nc1)C(=O)OCC

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.53
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9068196 0.86 DHFR (0.57) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL12692389 0.80 DHFR (0.55) DHFR
SCHEMBL9765081 0.79 DHFR (0.56) DHFR
SCHEMBL9765074 0.79 DHFR (0.56) DHFR
SCHEMBL10697242 0.79 DHFR (0.63) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL9313700 0.77 DHFR (0.69) DHFRKDM4EALDH1A1HPGDHSD17B10
SCHEMBL11439137 0.75 DHFR (0.65) DHFR
SCHEMBL10963943 0.75 DHFR (0.65) DHFR
SCHEMBL10963951 0.75 DHFR (0.65) DHFR
SCHEMBL8323452 0.75 DHFR (0.52) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536724-A Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins SRI INTERNATIONAL (US) 1996-07-16 US disclosed
EP-0638079-A1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1995-02-15 EP disclosed
WO-1993022312-A1 DEAZAAMINOPTERINS FOR TREATMENT OF INFLAMMATION SRI INTERNATIONAL (US) 1993-11-11 WO disclosed