SCHEMBL9765074

SCHEMBL9765074

CCOC(=O)CC[C@H](NC(=O)c1ccc(C(CC)Cc2cnc3nc(N)nc(N)c3c2C)cc1)C(=O)OCC

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.56
FOLR1 P15328 1/20 0.46
SLC19A1 P41440 1/20 0.46
SLC46A1 Q96NT5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765081 1.00 DHFR (0.56) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL9765067 0.87 DHFR (0.71) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL12692389 0.85 DHFR (0.55) DHFR
SCHEMBL10697242 0.84 DHFR (0.63) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL9540646 0.81 DHFR (0.45) DHFR
SCHEMBL9544497 0.80 DHFR (0.47) DHFR
SCHEMBL9068436 0.79 DHFR (0.53) DHFR
SCHEMBL8323452 0.78 DHFR (0.52) DHFR
SCHEMBL15075306 0.78 DHFR (0.75) DHFRFOLR1SLC19A1SLC46A1
SCHEMBL8323453 0.78 DHFR (0.52) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5077404-A Cyclized 5,10-dideazaaminopterin compounds SRI INTERNATIONAL 1991-12-31 US disclosed