SCHEMBL9073294

SCHEMBL9073294

C[C@]12CCC(=O)C=C1CC[C@@H]1C2=CC[C@]2(C)C(C(=O)CO)=CC[C@@H]12

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 17/20 0.63
NR3C1 P04150 1/20 0.52
CYP17A1 P05093 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10708164 0.91 CYP19A1 (0.62) CYP19A1NR3C1CYP17A1
SCHEMBL8999931 0.89 CYP19A1 (0.67) CYP19A1NR3C1CYP17A1
SCHEMBL2118371 0.88 NR3C1 (0.64) CYP19A1NR3C1CYP17A1
SCHEMBL8999936 0.88 NR3C1 (0.64) CYP19A1NR3C1CYP17A1
SCHEMBL9356635 0.86 CYP19A1 (0.56) CYP19A1NR3C1CYP17A1
SCHEMBL9356884 0.86 CYP19A1 (0.56) CYP19A1NR3C1CYP17A1
SCHEMBL9356926 0.84 CYP19A1 (0.54) CYP19A1NR3C1CYP17A1
SCHEMBL8668371 0.84 CYP19A1 (0.54) CYP19A1NR3C1CYP17A1
SCHEMBL9360771 0.84 CYP19A1 (0.53) CYP19A1NR3C1CYP17A1
SCHEMBL11332229 0.83 CYP19A1 (0.57) CYP19A1NR3C1CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0350488-B1 1,2-DEHYDROGENATION OF STEROIDAL 21-ESTERS WITH A. SIMPLEX THE UPJOHN COMPANY (US) 1993-09-08 EP claimed
EP-0350488-A1 1,2-DEHYDROGENATION OF STEROIDAL 21-ESTERS WITH A. SIMPLEX. UPJOHN CO (US) 1990-01-17 EP claimed
WO-1988007092-A1 1,2-DEHYDROGENATION OF STEROIDAL 21-ESTERS WITH A. SIMPLEX THE UPJOHN COMPANY (US) 1988-09-22 WO claimed
CN-116410939-A 3-sterone-delta 1 Dehydrogenase mutant and application thereof in synthesis of steroid C1,2 dehydrogenation drug intermediates 中国科学院天津工业生物技术研究所 2023-07-11 CN disclosed
US-5506354-A ANTIULCER, ANTITURMOR, ANTIARTHRITIC, ANTIATHEROSCLEROSIS, ANTIALLERGIC, ANTIASTHMA AGENTS THE UPJOHN COMPANY (US) 1996-04-09 US disclosed
EP-0238545-B1 C20 THROUGH C26 AMINO STEROIDS UPJOHN CO (US) 1995-11-15 EP disclosed
US-RE35053-E Intermediates for amino substituted steroids THE UPJOHN COMPANY (US) 1995-10-10 US disclosed
EP-0263213-B1 C20 Through C26 amino steroids UPJOHN CO (US) 1995-09-06 EP disclosed
US-5382661-A Useful in treating spinal trauma, head injury, subarachnoid hemorrhage THE UPJOHN COMPANY (US) 1995-01-17 US disclosed
US-5380841-A Steroids as antiinflammatory agents THE UPJOHN COMPANY (US) 1995-01-10 US disclosed
US-5380839-A Antitumor agents, antisecretory agents, enzyme inhibitors or antiasthmatics THE UPJOHN COMPANY (US) 1995-01-10 US disclosed
WO-1988007092-A1 1,2-DEHYDROGENATION OF STEROIDAL 21-ESTERS WITH A. SIMPLEX THE UPJOHN COMPANY (US) 1988-09-22 WO disclosed
EP-0263213-A1 C20 Through C26 amino steroids THE UPJOHN COMPANY (US) 1988-04-13 EP disclosed
US-4704455-A 16α-methylatedΔ17(20)-corticoids THE UPJOHN COMPANY (US) 1987-11-03 US disclosed
EP-0238545-A1 C 20? THROUGH C 26? AMINO STEROIDS. UPJOHN CO (US) 1987-09-30 EP disclosed
WO-1987001706-A2 C20 THROUGH C26 AMINO STEROIDS THE UPJOHN COMPANY (US) 1987-03-26 WO disclosed
EP-0175540-A2 20-Silyl ether steroids, and preparing 17-hydroxy-20-keto steroids THE UPJOHN COMPANY (US) 1986-03-26 EP disclosed
US-4568492-A HYDROSILYLATION THEN PERACID OXIDATION THE UPJOHN COMPANY (US) 1986-02-04 US disclosed
EP-0127216-A1 Process for the preparation of 21-hydroxy-20-keto-delta16-steroids and intermediate compounds formed in this process ROUSSEL-UCLAF (FR) 1984-12-05 EP disclosed
EP-0123736-A1 New process for the preparation of 21-hydroxy-20-keto-delta 16-steroids and new intermediate compounds formed in this process GIST-BROCADES N.V. (NL) 1984-11-07 EP disclosed