SCHEMBL9074615

SCHEMBL9074615

Cc1cccc(CBr)c1C(=O)OO[Si](C)(C)C(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.33
PREP P48147 2/20 0.32
MAOB P27338 2/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA7 P43166 1/20 0.30
CA9 Q16790 1/20 0.30
CA14 Q9ULX7 1/20 0.30
POLB P06746 1/20 0.30
ELANE P08246 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9075036 0.85 TDP1 (0.33) CA12CA1CA2CA7CA9
SCHEMBL28360772 0.79 CA12 (0.37) MAOBCA12CA1CA2CA7
SCHEMBL3093326 0.79 GRM6 (0.39) CA12CA1CA2CA7CA9
SCHEMBL2876253 0.76 CA12 (0.48) CA12CA1CA2CA7CA9
SCHEMBL5693160 0.75 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL5837073 0.74 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL15129901 0.73 HDAC1 (0.43) BACE1PREPCA12CA1CA2
SCHEMBL9070648 0.72 ADRB2 (0.46) MAPT
SCHEMBL2879882 0.72 SCN4A (0.35) PREPPOLBELANEALDH1A1
SCHEMBL4841311 0.71 ALDH1A1 (0.50) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486466-A ENZYME INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1996-01-23 US disclosed
US-5399741-A DNA gyrase inhibitors, process for their manufacture and pharmaceutical preparations containing same HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
EP-0535192-A1 NOVEL DNA GYRASE INHIBITORS, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL PREPARATIONS CONTAINING SAME. HOFFMANN LA ROCHE (CH) 1993-04-07 EP disclosed