SCHEMBL9079302

SCHEMBL9079302

CC(O)=C(C#N)C(=O)Nc1ccc(Oc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.85

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 8/20 0.85
FNTA P49354 1/20 0.46
FNTB P49356 1/20 0.46
EPHX2 P34913 1/20 0.44
TRPV1 Q8NER1 2/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
BRAF P15056 1/20 0.43
KDR P35968 1/20 0.43
MAPK14 Q16539 1/20 0.43
TNNI3K Q59H18 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8808801 1.00 DHODH (0.85) DHODHFNTAFNTBEPHX2TRPV1
Teriflunomide SCHEMBL22661 0.92 DHODH (1.00) DHODHEPHX2TRPV1
Teriflunomide SCHEMBL993119 0.92 DHODH (1.00) DHODHEPHX2TRPV1
Teriflunomide SCHEMBL20214092 0.92 DHODH (1.00) DHODHEPHX2TRPV1
Teriflunomide SCHEMBL2760666 0.92 DHODH (1.00) DHODHEPHX2TRPV1
Teriflunomide SCHEMBL991312 0.91 DHODH (0.97) DHODHEPHX2TRPV1
Teriflunomide SCHEMBL8466730 0.91 DHODH (0.97) DHODHEPHX2TRPV1
Teriflunomide SCHEMBL992140 0.91 DHODH (0.97) DHODHEPHX2TRPV1
SCHEMBL9178600 0.88 DHODH (0.66) DHODHFNTAFNTBEPHX2TRPV1
SCHEMBL9081065 0.87 DHODH (0.64) DHODHFNTAFNTBEPHX2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5532259-A ANTITUMOR HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-02 US disclosed
US-5494911-A TREATING LEUKEMIA, SARCOMA, CARCINOMA, LYMPHOMA, SKIN CANCER HOECHST AKTIENGESELLSCHAFT (DE) 1996-02-27 US disclosed